{"id":23662,"date":"2025-04-13T17:40:11","date_gmt":"2025-04-13T17:40:11","guid":{"rendered":"https:\/\/researchchemworld.com\/?post_type=product&#038;p=23662"},"modified":"2026-02-26T13:24:39","modified_gmt":"2026-02-26T13:24:39","slug":"flualprazolam-1-mg-pelety","status":"publish","type":"product","link":"https:\/\/researchchemworld.com\/cs\/nakupovat\/zakazano\/flualprazolam-1-mg-pelety\/","title":{"rendered":"Flualprazolam 1 MG pelety"},"content":{"rendered":"<div id=\"content_tab_description\" class=\"tab-content tab-description\">\n<div class=\"tab-content-inner\">\n<div class=\"tab-content-scroll\">\n<h1><strong>Flualprazolam 1 mg pelety \u2013 v\u00fdzkumn\u00e1 slou\u010denina se silnou benzodiazepinovou aktivitou<\/strong><\/h1>\n<p><strong>N\u00e1zev produktu:<\/strong> Flualprazolam 1 MG pelety<br \/>\n<strong>Chemick\u00e1 t\u0159\u00edda:<\/strong> Triazolobenzodiazepiny<br \/>\n<strong>Vzorec:<\/strong> C17H12ClFN4<br \/>\n<strong>Molekulov\u00e1 hmotnost:<\/strong> 342,8 g\/mol<br \/>\n<strong>\u010cistota:<\/strong> \u2265 98% (ov\u011b\u0159eno HPLC)<br \/>\n<strong>Formul\u00e1\u0159:<\/strong> Mikrolisovan\u00e9 pelety o hmotnosti 1 mg<\/p>\n<hr \/>\n<h2><strong>Popis<\/strong><\/h2>\n<p>Flualprazolam je siln\u00e1 slou\u010denina ze t\u0159\u00eddy benzodiazepin\u016f, strukturn\u011b podobn\u00e1 alprazolamu (Xanax), jeho\u017e charakteristick\u00fdm znakem je p\u0159id\u00e1n\u00ed atomu fluoru k fenylov\u00e9mu kruhu. Tato jemn\u00e1 chemick\u00e1 modifikace zvy\u0161uje afinitu k receptor\u016fm GABAA, co\u017e vede ke zv\u00fd\u0161en\u00e9 \u00fa\u010dinnosti a del\u0161\u00edmu trv\u00e1n\u00ed \u00fa\u010dinku.<\/p>\n<p>Pelety Flualprazolamu 1 mg jsou p\u0159esn\u011b d\u00e1vkovan\u00e9 a ur\u010den\u00e9 v\u00fdhradn\u011b pro <strong>analytick\u00e9 \u00fa\u010dely, referen\u010dn\u00ed v\u00fdzkum a laboratorn\u00ed anal\u00fdza<\/strong>Nen\u00ed ur\u010deno k lidsk\u00e9 spot\u0159eb\u011b.<\/p>\n<hr \/>\n<h2><strong>Aplikace a v\u00fdzkumn\u00e9 \u00fa\u010dely<\/strong><\/h2>\n<ul>\n<li>Farmakodynamick\u00e9 studie GABAergn\u00edch interakc\u00ed<\/li>\n<li>Studie vazby na receptory a srovn\u00e1n\u00ed s jin\u00fdmi triazolobenzodiazepiny<\/li>\n<li>Behavior\u00e1ln\u00ed studie na zv\u00ed\u0159ec\u00edch modelech za kontrolovan\u00fdch podm\u00ednek<\/li>\n<li>Anal\u00fdzy stability a rozpustnosti v r\u016fzn\u00fdch rozpou\u0161t\u011bdlech<\/li>\n<li>Referen\u010dn\u00ed \u00fadaje v toxikologick\u00fdch nebo analytick\u00fdch laborato\u0159\u00edch (kalibrace GC-MS\/LC-MS)<\/li>\n<\/ul>\n<hr \/>\n<h2><strong>V\u00fdhody pro v\u00fdzkumn\u00edky<\/strong><\/h2>\n<p>\u2705 <strong>Vysok\u00e1 \u00fa\u010dinnost<\/strong> \u2013 Pro znateln\u00e9 \u00fa\u010dinky v experiment\u00e1ln\u00edm prost\u0159ed\u00ed je nutn\u00e1 n\u00edzk\u00e1 d\u00e1vka<br \/>\n\u2705 <strong>Stabiln\u00ed tvar pelet<\/strong> \u2013 Snadn\u00e9 d\u00e1vkov\u00e1n\u00ed a skladov\u00e1n\u00ed<br \/>\n\u2705 <strong>Laboratorn\u011b testovan\u00e1 \u010distota<\/strong> \u2013 Zaru\u010dena konzistence pro reprodukovateln\u00e9 v\u00fdsledky v\u00fdzkumu<\/p>\n<hr \/>\n<h2><strong>Nev\u00fdhody a rizika<\/strong><\/h2>\n<p>\u26a0\ufe0f <strong>Velmi siln\u00fd<\/strong> \u2013 I nepatrn\u00e9 odchylky v d\u00e1vkov\u00e1n\u00ed mohou v\u00fdrazn\u011b ovlivnit v\u00fdsledek experiment\u016f<br \/>\n\u26a0\ufe0f <strong>Dlouhotrvaj\u00edc\u00ed \u00fa\u010dinek<\/strong> \u2013 M\u016f\u017ee v\u00e9st k akumulaci u zv\u00ed\u0159ec\u00edch model\u016f po opakovan\u00e9m pod\u00e1n\u00ed<br \/>\n\u26a0\ufe0f <strong>Pot\u0159eba podm\u00edn\u011bn\u00e9ho skladov\u00e1n\u00ed<\/strong> \u2013 Skladujte nejl\u00e9pe p\u0159i teplot\u011b do 25 \u00b0C, v suchu a tm\u011b<\/p>\n<hr \/>\n<h2><strong>Pou\u017eit\u00ed a laboratorn\u00ed pokyny<\/strong><\/h2>\n<ul>\n<li><strong>Doporu\u010den\u00e9 laboratorn\u00ed d\u00e1vkov\u00e1n\u00ed:<\/strong> Pro in vitro testy za\u010dn\u011bte s d\u00e1vkou 0,25\u20130,5 mg. Bez kalibrace nep\u0159ekra\u010dujte tuto d\u00e1vku.<\/li>\n<li><strong>Rozpustnost:<\/strong> Voln\u011b rozpustn\u00fd v ethanolu, DMSO a propylenglykolu<\/li>\n<li><strong>Podm\u00ednky skladov\u00e1n\u00ed:<\/strong> Skladujte ve vzduchot\u011bsn\u00e9 n\u00e1dob\u011b, v chladu a mimo dosah p\u0159\u00edm\u00e9ho slune\u010dn\u00edho z\u00e1\u0159en\u00ed<\/li>\n<li><strong>Zach\u00e1zen\u00ed:<\/strong> P\u0159i manipulaci s pr\u00e1\u0161kem nebo roztokem pou\u017e\u00edvejte rukavice, ochrann\u00e9 br\u00fdle a pracujte pod digesto\u0159\u00ed.<\/li>\n<\/ul>\n<hr \/>\n<h2><strong>\u010casto kladen\u00e9 ot\u00e1zky (FAQ)<\/strong><\/h2>\n<h3>\u2753 <em>Je Flualprazolam leg\u00e1ln\u00ed v Nizozemsku nebo Belgii?<\/em><\/h3>\n<p>\u27a1\ufe0f Pr\u00e1vn\u00ed status se li\u0161\u00ed. V\u017edy si ov\u011b\u0159te nejnov\u011bj\u0161\u00ed m\u00edstn\u00ed p\u0159edpisy. Konzumace je obecn\u011b zak\u00e1z\u00e1na, ale m\u016f\u017ee b\u00fdt povolena pro analytick\u00e9 testy.<\/p>\n<h3>\u2753 <em>Mohu Flualprazolam pou\u017e\u00edvat k v\u00fdzkumu sp\u00e1nku nebo \u00fazkosti?<\/em><\/h3>\n<p>\u27a1\ufe0f Pouze v p\u0159\u00edsn\u011b kontrolovan\u00e9m laboratorn\u00edm prost\u0159ed\u00ed a v\u00fdhradn\u011b na nelidsk\u00fdch modelech nebo ve studi\u00edch chemick\u00fdch interakc\u00ed.<\/p>\n<h3>\u2753 <em>Jak dlouho z\u016fst\u00e1v\u00e1 flualprazolam stabiln\u00ed p\u0159i pokojov\u00e9 teplot\u011b?<\/em><\/h3>\n<p>\u27a1\ufe0f V suchu a tm\u011b z\u016fst\u00e1v\u00e1 stabiln\u00ed po dobu nejm\u00e9n\u011b 12 m\u011bs\u00edc\u016f p\u0159i teplot\u011b 20\u201325 \u00b0C.<\/p>\n<h3>\u2753 <em>Existuje zk\u0159\u00ed\u017een\u00e1 rezistence s jin\u00fdmi benzodiazepiny?<\/em><\/h3>\n<p>\u27a1\ufe0f Ano, flualprazolam vykazuje p\u0159ekr\u00fdvaj\u00edc\u00ed se vazebn\u00e9 profily s jin\u00fdmi l\u00e1tkami, jako je alprazolam a klonazolam.<\/p>\n<hr \/>\n<h2><strong>Shrnut\u00ed laboratorn\u00ed zpr\u00e1vy<\/strong><\/h2>\n<table>\n<thead>\n<tr>\n<th>Parametr<\/th>\n<th>Hodnota<\/th>\n<\/tr>\n<\/thead>\n<tbody>\n<tr>\n<td><strong>\u010c\u00edslo \u0161ar\u017ee<\/strong><\/td>\n<td>FLPZ-0725<\/td>\n<\/tr>\n<tr>\n<td><strong>\u010cistota (HPLC)<\/strong><\/td>\n<td>99,3%<\/td>\n<\/tr>\n<tr>\n<td><strong>Vzhled<\/strong><\/td>\n<td>B\u00edl\u00fd krystalick\u00fd pr\u00e1\u0161ek (slisovan\u00fd do pelet)<\/td>\n<\/tr>\n<tr>\n<td><strong>Bod t\u00e1n\u00ed<\/strong><\/td>\n<td>225\u2013230 \u00b0C<\/td>\n<\/tr>\n<tr>\n<td><strong>Identifikace<\/strong><\/td>\n<td>Potvrzeno NMR a MS<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<hr \/>\n<h2><strong>Varov\u00e1n\u00ed<\/strong><\/h2>\n<p><strong>Nen\u00ed ur\u010deno k lidsk\u00e9 spot\u0159eb\u011b ani k l\u00e9ka\u0159sk\u00e9mu pou\u017eit\u00ed. Pouze pro profesion\u00e1ln\u00ed v\u00fdzkum v kvalifikovan\u00fdch laborato\u0159\u00edch.<\/strong><\/p>\n<\/div>\n<\/div>\n<\/div>","protected":false},"excerpt":{"rendered":"<h3><span data-sheets-value=\"{\" data-sheets-userformat=\"{\"><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Flualprazolam Pellets Properties<\/span><\/span><\/span><\/h3>\n<p><strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Synonym:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> Fluclazolam <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">CAS Number:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> 28910-91-0 <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Formula:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> 8-chloro-6-(2-fluorophenyl)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Molar mass:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> 326.8 g\/mol <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Purity:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> &gt;97%<\/span><\/span><\/p>\n","protected":false},"featured_media":29349,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[488],"product_tag":[326],"class_list":{"0":"post-23662","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-verboden","7":"product_tag-nl","9":"first","10":"instock","11":"taxable","12":"shipping-taxable","13":"purchasable","14":"product-type-simple"},"_links":{"self":[{"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/product\/23662","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/comments?post=23662"}],"version-history":[{"count":4,"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/product\/23662\/revisions"}],"predecessor-version":[{"id":25752,"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/product\/23662\/revisions\/25752"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/media\/29349"}],"wp:attachment":[{"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/media?parent=23662"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/product_brand?post=23662"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/product_cat?post=23662"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/researchchemworld.com\/cs\/wp-json\/wp\/v2\/product_tag?post=23662"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}