{"id":23116,"date":"2025-04-13T17:39:10","date_gmt":"2025-04-13T17:39:10","guid":{"rendered":"https:\/\/researchchemworld.com\/?post_type=product&#038;p=23116"},"modified":"2026-02-26T15:45:14","modified_gmt":"2026-02-26T15:45:14","slug":"etisolaami-1-mg-graanulid","status":"publish","type":"product","link":"https:\/\/researchchemworld.com\/et\/pood\/keelatud\/etisolaami-1-mg-graanulid\/","title":{"rendered":"Etizolam 1 MG graanulid"},"content":{"rendered":"<h1><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolam 1 MG pelletid \u2013 tienodiazepiini laboratoorse kvaliteediga uurimisvorm<\/span><\/span><\/strong><\/h1>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolami \u00fclevaade<\/span><\/span><\/h2>\n<p><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etisolaam on tienodiazepiini analoog, millel on tugevad anksiol\u00fc\u00fctilised, rahustavad ja lihaseid l\u00f5\u00f5gastavad omadused. Need 1 mg graanulid t\u00f6\u00f6tati v\u00e4lja GABA-A retseptorite interaktsioonide ja neurofarmakoloogiliste protsesside kontrollitud uuringuteks. <\/span><\/span><a href=\"https:\/\/researchchemworld.com\/et\/pood\/lusergamiidid\/1vlsd\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">1V-LSD 150 MCG blotterid<\/span><\/span><\/a><\/p>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Toote omadused<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">T\u00e4pselt 1 mg etisolaami pelleti kohta (\u00b12% variatsioon)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Mikrokristalse tselluloosiga valmistatud<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Fotostabiilne ja niiskuskindel pakend<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Partii kontrolliti j\u00e4rgmiste n\u00e4itajate suhtes:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">HPLC puhtus (\u226598%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">MS-i identiteedi kontrollimine<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Kaalu ja suuruse \u00fchtlus<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Farmakoloogiline profiil<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">K\u00f5rge afiinsus GABA-A retseptorite suhtes<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Selektiivne seondumine \u03b11\u2013\u03b15 alat\u00fc\u00fcpidega<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Farmakoloogiline toime:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Anksiol\u00fc\u00fctikum<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Rahustav<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Lihasrelaksant<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">L\u00fchem eliminatsiooni poolv\u00e4\u00e4rtusaeg kui klassikalistel bensodiasepiinidel<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Rakendusvaldkonnad uurimist\u00f6\u00f6s<\/span><\/span><\/h2>\n<ol>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Neurofarmakoloogia<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">GABA-A retseptori interaktsioonid<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Allosteeriline modulatsioon<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Alamt\u00fc\u00fcbi spetsiifilisus<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">V\u00f5rdlev anal\u00fc\u00fcs<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Struktuuri ja aktiivsuse v\u00f5rdlus bensodiasepiinidega<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Ainevahetusradade uuringud<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">K\u00e4itumisteadus<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u00c4revusmudelid (nt EPM, OFT)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Une- ja \u00e4rkveloleku ts\u00fcklid<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Krampide p\u00e4rssimine<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ol>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Tehnilised andmed<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Pelleti l\u00e4bim\u00f5\u00f5t: 2,5 mm \u00b1 0,1 mm<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Kaal: 10 mg \u00b1 0,5 mg<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">V\u00e4rv: Puhas valge<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Lahustuvus: &gt;5 mg\/ml etanoolis (96%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Sulamistemperatuur: 146\u2013148 \u00b0C<\/span><\/span><\/li>\n<\/ul>\n<h3><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Stabiilsusprofiil<\/span><\/span><\/h3>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">S\u00e4ilivusaeg: 36 kuud temperatuuril 15\u201325 \u00b0C<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Valguskindlus: &lt;1% lagunemine\/aasta<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Niiskusesisaldus: &lt;0,5% (Karl Fischer)<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Annustamisjuhised (ainult viitamiseks)<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">In vitro: 10\u20131000 nM<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Prekliiniline: 0,05\u20130,5 mg\/kg<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">K\u00e4itumismudelid: 0,1\u20131,0 mg\/kg<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Ohutus- ja hoiustamisteave<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Hoida valgusekindlas pakendis<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Suhteline \u00f5huniiskus &lt;40%<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Temperatuur vahemikus 15\u201325 \u00b0C<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">\u00dchildub PBS-i ja NaCl 0,9%-ga <\/span><\/span><a href=\"https:\/\/researchchemworld.com\/et\/pood\/pellets\/o-dsmt-50mg-graanulid\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">O-DSMT 50 mg graanulid<\/span><\/span><\/a><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Dokumentatsioon kohaletoimetamisel<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Autentsussertifikaat koos:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Puhtus<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">S\u00e4ilitusaeg<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Massiline identifitseerimine<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Ohutuskaart (SDS) vastavalt GHS-ile<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Tehniline leht koos:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Stabiilsusandmed<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Eksperimentaalse disaini ettepanekud<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Lahustuvuse anal\u00fc\u00fcs<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<p><em><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Ainult teaduslikul eesm\u00e4rgil. Ei sobi meditsiiniliseks, diagnostiliseks ega inimtoiduks. <\/span><\/span><a href=\"https:\/\/researchchemworld.com\/et\/pood\/top-10-research-chemicals\/caluanie-muelear-oksudeerub\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Caluanie Muelear Oxidize<\/span><\/span><\/a><\/em><\/p>","protected":false},"excerpt":{"rendered":"<h2><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolam pellets properties<\/span><\/span><\/span><\/span><\/h2>\n<p><strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Synonym<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 4-(2-chlorophenyl)-2-ethyl-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">CAS Number<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 40054-69-1 <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Formula<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : C17H15ClN4S <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Molar mass<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 342.8 g\/mol <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Purity<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : \u2265 99%<\/span><\/span><\/span><\/span><\/p>\n","protected":false},"featured_media":29344,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[82],"product_cat":[488],"product_tag":[917,326],"class_list":{"0":"post-23116","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_brand-research-chemical","7":"product_cat-verboden","8":"product_tag-etizolam","9":"product_tag-nl","11":"first","12":"instock","13":"taxable","14":"shipping-taxable","15":"purchasable","16":"product-type-simple"},"_links":{"self":[{"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/product\/23116","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/comments?post=23116"}],"version-history":[{"count":6,"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/product\/23116\/revisions"}],"predecessor-version":[{"id":28492,"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/product\/23116\/revisions\/28492"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/media\/29344"}],"wp:attachment":[{"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/media?parent=23116"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/product_brand?post=23116"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/product_cat?post=23116"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/researchchemworld.com\/et\/wp-json\/wp\/v2\/product_tag?post=23116"}],"curies":[{"name":"t\u00f6\u00f6leht","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}