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Etizolam 1 mg mikro peleti

Lastnosti mikro peletov Etizolama

Sinonim 4-(2-klorofenil)-2-etil-9-metil-6H-tieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin
Številka CAS : 40054-69-1
Formula C17H15ClN4S
Molska masa : 342,8 g/mol
Čistost : ≥ 99%

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Etizolam 1 MG Micro Pellets – Precision Dosing for Research Purposes

Product Name: Etizolam 1 mg mikro pelete
Active Substance: Etizolam
Chemical Class: Thienodiazepine (benzodiazepine analogue)
Molekularna formula: C17H15ClN4S
Molecular Mass: 342.85 g/mol
Oblika: Micro Pellets (submillimeter size)
Odmerjanje: 1 mg na peleto
Packaging: 10 / 25 / 50 / 100 peletov
Application: For laboratory and analytical research only


🔬 What is Etizolam?

Etizolam is a thienodiazepine compound structurally related to traditional benzodiazepines. It is known for its potent GABA-A receptor agonism , which produces anxiolytic, sedative, and muscle relaxant effects . In analytical studies, Etizolam is being evaluated for its receptor binding profile , stability , and structural-activity relationships (SAR) within the benzodiazepine family.

The micro pellet shape offers exceptional precision dosing and reproducibility , ideal for fine-mesh laboratory applications and storage.


Uporaba v raziskavah

  • Neuroreceptor analysis: GABA-A modulation in vitro
  • Structural activity study (SAR): Comparison with classical benzos (diazepam, alprazolam)
  • Stability studies: Under the influence of temperature, moisture and light
  • Pharmacokinetics (preclinical): In vivo simulations under ethical protocol
  • Analytical reference substance: LC-MS, HPLC, NMR

⚠️ Pozor: Not suitable for human or animal consumption. For professional research purposes only.


⚠️ Risks and Limitations

  • Very potent in low doses – incorrect use can be dangerous
  • Dependency potential with abuse
  • Possible regulation in EU/US – considered a controlled substance in some countries
  • Not intended for recreational use or self-experimentation
  • May cause drowsiness or motor disorders if handled incorrectly

🧪 Laboratory details

CharacteristicSpecification
Active substanceEtizolam (≥99% purity – HPLC, GC-MS)
FormMicro pellets (approximately 0.6–0.8 mm diameter)
Odmerjanje1 mg na peleto
ColourWhite to light gray
Stabilnost≥ 24 months when stored correctly
SolubilitySoluble in ethanol, DMSO, acetonitrile
Nasveti za shranjevanjeDark, dry, cool (2–8 °C)
potrdilo o avtornostiAvailable upon request

💡 Recommended Use Cases

Research areaApplication
Študije vezave receptorjevGABA-A response in different subtypes
Analitska kemijaReference in HPLC or LC-MS equipment
Stability testingUnder stressful conditions in the laboratory
Raziskave SARComparison with other thienodiazepines

Pogosto zastavljena vprašanja (FAQ)

1. What is the difference between a micro pellet and a regular pellet?
Micro pellets are much smaller (submillimeter size) and designed for highly accurate dosing and rapid dissolution during analytical processes.

2. Is Etizolam legal?
That varies by country. In some regions, Etizolam is a controlled substance . Always check the regulations in your country before ordering or using it.

3. Is this product suitable for human consumption?
No. These pellets are intended for laboratory use only . Use on humans or animals is prohibited and potentially dangerous.

4. How should I store the pellets?
Store them in a tightly closed, dry container at 2–8°C , protected from light and moisture.

5. Is a Certificate of Analysis available?
Yes, a COA (Potrdilo o analizi) is available upon request for each batch. This includes HPLC data, purity, and lot number.


📦 Product overview

FeatureSpecification
Product nameEtizolam 1 mg mikro peleti
FormSubmillimeter pressed pellets
Odmerjanje1 mg na peleto
Embalaža10 / 25 / 50 / 100 peletov
Čistost≥99%
UsageFor laboratory use only
Storage conditionCool, dry, light-free
Legal statusRegion dependent
potrdilo o avtornostiAvailable per batch

 

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